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Search Results for " a-3 hydrochloride "

20

Compounds

Cat No. Product Name Synonyms Targets
T14069 A-3 hydrochloride CaMK , Casein Kinase , PKA , PKC
A-3 hydrochloride is a potent, cell-permeable, reversible, ATP-competitive non-selective antagonist of various kinases. A-3 hydrochloride also inhibits PKC and casein kinase I with Ki values of 47 µM and 80 µM, respectiv...
T9881 Benzoquinamide hydrochloride 3-carbamoyl-N,N-diethyl-1,3,4,6,7,11b-hexahydro-9,11-dimethoxy-2H-benzo[a]quinolizin-2-yl acetate hydrochloride Others
Benzoquinamide hydrochloride (3-carbamoyl-N,N-diethyl-1,3,4,6,7,11b-hexahydro-9,11-dimethoxy-2H-benzo[a]quinolizin-2-yl acetate hydrochloride) is an antiemetic agent and increases intra-arterial pressure due to the incre...
T2287 PIK-75 hydrochloride PIK-75 HCl,PIK-75 Apoptosis , DNA-PK , PI3K
PIK-75 hydrochloride (PIK-75 HCl) is a p110α inhibitor with IC50 of 5.8 nM (200-fold more potently than p110β), isoform-specific mutants at Ser773, and also potently inhibits DNA-PK with IC50 of 2 nM in cell-free assays.
T35526 PI3-Kinase α Inhibitor 2 (hydrochloride) PI3-Kinase α Inhibitor 2 (hydrochloride)
PI3-Kinase α Inhibitor 2 (hydrochloride) is a PI3-Kinase α inhibitor.
T5978 2,3-Diaminopropionic acid hydrochloride 3-Amino-L-alanine hydrochloride Others
2,3-Diaminopropionic acid hydrochloride (3-Amino-L-alanine hydrochloride) is a competitive cystathionase(CTH) inhibitor.
T5683 (2R,3S)-3-Phenylisoserine hydrochloride Others
"(2R,3S)-3-Phenylisoserine hydrochloride serves as a pharmaceutical intermediate."
T12906 SI-2 hydrochloride EPH 116 hydrochloride Src
SI-2 hydrochloride (EPH 116 hydrochloride) is a highly promising inhibitor of SRC-3 SMI: SRC-3 (PPI)(IC50 values of 3-20 nM for breast cancer cell death), with acceptable oral availability.
T11188L Emixustat hydrochloride ACU-4429 hydrochloride Others
Emixustat hydrochloride (ACU-4429 hydrochloride) strongly inhibits 11-cis-retinol production with IC50 values of 232 ± 3 nM. 11-cis-retinol Emixustat hydrochloride is a novel visual cycle modulator.
T61972 Pomaglumetad methionil hydrochloride LY2140023 hydrochloride GluR
Pomaglumetad methionine hydrochloride (LY2140023 hydrochloride) is a methionine prodrug of LY404039 with oral activity. LY404039 is a selective mGlu2/3 receptor agonist. Pomaglumetad methionil hydrochloride (LY2140023 hy...
T4710 3-Methoxytyramine hydrochloride 3-O-methyl Dopamine hydrochloride,3-O-methyl Dopamine hydrochloride) Others , Endogenous Metabolite , Drug Metabolite
3-Methoxytyramine hydrochloride (3-O-methyl Dopamine hydrochloride) is an inactive metabolite of dopamine which can activate trace amine associated receptor 1 (TAAR1). 3-methoxytyramine can be found primarily in human br...
T10394L ATB107 hydrochloride ATB107 hydrochloride(455325-51-6 Free base) Others
ATB107 hydrochloride is a novel and potent inhibitor of indole-3-glycerol phosphate synthase (IGPS) with a KD of 3 μM.
T4234 HJC0152 hydrochloride HJC0152 Apoptosis , STAT
HJC0152 hydrochloride (HJC0152) is a signal transducer and activator of transcription 3 (STAT3) inhibitor.
T8494 NS-3-008 hydrochloride NS-3-008 HCl Others
NS-3-008 hydrochloride (NS-3-008 HCl) is a transcriptional G0/G1 switch 2 (G0s2) inhibitor( IC50 of 2.25 μM).
T40031 Thalidomide-O-C6-NH2 hydrochloride 4-((6-aminohexyl)oxy)-2-(2,6-dioxopiperidin-3-yl)isoindoline-1,3-dione hydrochloride E3 Ligase Ligand-Linker Conjugate
Thalidomide-O-C6-NH2 hydrochloride (4-((6-aminohexyl)oxy)-2-(2,6-dioxopiperidin-3-yl)isoindoline-1,3-dione hydrochloride) is a synthesized E3 ligase ligand-linker conjugate.
T22638 CBiPES hydrochloride CBiPES HCl GluR
CBiPES hydrochloride (CBiPES HCl) is a potent orthosteric modulator of the mGlu2 receptor with an EC50 value of 92.8 nM.CBiPES hydrochloride blocks the action of WT and mGlu(3) receptors.CBiPES hydrochloride can be used ...
T12930 SKF89976A hydrochloride d,l-SKF89976A hydrochloride GABA Receptor
SKF89976A hydrochloride (d,l-SKF89976A hydrochloride) is a selective inhibitor GABA transporter such as GAT-1 (IC50s = 0.28 μM), GAT-2 (IC50s = 137.34 μM) and GAT-3(IC50s = 202.8 μM) in CHO cells.
T11638 Ilorasertib hydrochloride ABT-348 hydrochloride Aurora Kinase
Ilorasertib hydrochloride (ABT-348 hydrochloride) is an ATP-competitive multitargeted kinase inhibitor, which inhibits Aurora C, Aurora B, and Aurora A (IC50s: 1 nM, 7 nM, 120 nM). It also suppresses RET tyrosine kinase,...
T4755 2,3-Diaminopropanoic acid hydrochloride DL-2,3-Diaminopropionic acid monohydroch,3-Amino-DL-alanine monohydrochloride Others , Endogenous Metabolite
2,3-Diaminopropanoic acid hydrochloride (3-Amino-DL-alanine monohydrochloride) is an amino acid amide used as a substrate for studying the action of aminopeptidase enzyme.
T1173 Tropisetron hydrochloride SDZ-ICS 930,Tropisetron HCl,ICS 205-930 5-HT Receptor
Tropisetron hydrochloride (Tropisetron HCl) is the hydrochloride salt form of tropisetron, a selective, competitive serotonin 5-hydroxytryptamine type 3 (5-HT3) receptor antagonist, with antinauseant and antiemetic activ...
T8639 Phenibut (hydrochloride) 3-Amino-4-phenylbutyric acid hydrochloride GABA Receptor
Phenibut hydrochloride (3-Amino-4-phenylbutyric acid hydrochloride) is a GABA mimetic that acts as an agonist at GABAB receptors, blocks α2δ subunit-containing voltage-gated calcium channels, stimulates dopamine receptor...

Compounds

A-3 hydrochloride
T14069
Synonym:
Target: CaMK, Casein Kinase, PKA, PKC
Benzoquinamide hydrochloride
T9881
Synonym: 3-carbamoyl-N,N-diethyl-1,3,4,6,7,11b-hexahydro-9,11-dimethoxy-2H-benzo[a]quinolizin-2-yl acetate hydrochloride
Target: Others
PIK-75 hydrochloride
T2287
Synonym: PIK-75 HCl,PIK-75
Target: Apoptosis, DNA-PK, PI3K
PI3-Kinase α Inhibitor 2 (hydrochloride)
T35526
Synonym: PI3-Kinase α Inhibitor 2 (hydrochloride)
Target:
2,3-Diaminopropionic acid hydrochloride
T5978
Synonym: 3-Amino-L-alanine hydrochloride
Target: Others
(2R,3S)-3-Phenylisoserine hydrochloride
T5683
Synonym:
Target: Others
SI-2 hydrochloride
T12906
Synonym: EPH 116 hydrochloride
Target: Src
Emixustat hydrochloride
T11188L
Synonym: ACU-4429 hydrochloride
Target: Others
Pomaglumetad methionil hydrochloride
T61972
Synonym: LY2140023 hydrochloride
Target: GluR
3-Methoxytyramine hydrochloride
T4710
Synonym: 3-O-methyl Dopamine hydrochloride,3-O-methyl Dopamine hydrochloride)
Target: Others, Endogenous Metabolite, Drug Metabolite
ATB107 hydrochloride
T10394L
Synonym: ATB107 hydrochloride(455325-51-6 Free base)
Target: Others
HJC0152 hydrochloride
T4234
Synonym: HJC0152
Target: Apoptosis, STAT
NS-3-008 hydrochloride
T8494
Synonym: NS-3-008 HCl
Target: Others
Thalidomide-O-C6-NH2 hydrochloride
T40031
Synonym: 4-((6-aminohexyl)oxy)-2-(2,6-dioxopiperidin-3-yl)isoindoline-1,3-dione hydrochloride
Target: E3 Ligase Ligand-Linker Conjugate
CBiPES hydrochloride
T22638
Synonym: CBiPES HCl
Target: GluR
SKF89976A hydrochloride
T12930
Synonym: d,l-SKF89976A hydrochloride
Target: GABA Receptor
Ilorasertib hydrochloride
T11638
Synonym: ABT-348 hydrochloride
Target: Aurora Kinase
2,3-Diaminopropanoic acid hydrochloride
T4755
Synonym: DL-2,3-Diaminopropionic acid monohydroch,3-Amino-DL-alanine monohydrochloride
Target: Others, Endogenous Metabolite
Tropisetron hydrochloride
T1173
Synonym: SDZ-ICS 930,Tropisetron HCl,ICS 205-930
Target: 5-HT Receptor
Phenibut (hydrochloride)
T8639
Synonym: 3-Amino-4-phenylbutyric acid hydrochloride
Target: GABA Receptor
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TargetMol